— COPPER-BINDING TRIPEPTIDE · WOUND & SKIN BIOREGULATOR

GHK-Cu.

A copper-chelating tripeptide found naturally in human plasma, saliva, and wound fluid. Studied across skin repair, hair regrowth, and tissue regeneration for over five decades — one of the most researched endogenous peptides in cosmetic and wound biology.

Key Signals
Collagen · Wound · Hair
Origin
Endogenous (human plasma)
Investigator
Loren Pickart, 1973
Class
Copper-binding tripeptide
Status (UAE)
Research compound (off-label)
— THE RESEARCH STORY

The Wound Healer Hidden in Plain Sight

Pickart identifies GHK as a plasma tripeptide that restores youthful liver function in aged tissue samples — 1973.

The Cu²⁺ chelation mechanism is characterised — enabling cuproenzyme activation critical to wound healing.

Adopted in cosmetic formulations globally; small human trials confirm collagen upregulation and elasticity gains.

— COLLAGEN SYNTHESIS RESPONSE
CONCEPTUAL · FIBROBLAST IN VITRO MODEL
100% 125% 155% 190% DAY 0 DAY 7 DAY 14 DAY 21 DAY 30
GHK-Cu TREATED UNTREATED CONTROL
— THE MOLECULE

A tripeptide with a copper payload

PRIMARY STRUCTURE

Gly · His · Lys · Cu²⁺

C₁₄H₂₃CuN₆O₄ · MW 340.8 Da

340.8MOLECULAR WEIGHT Da
3AMINO ACIDS
50+YEARS IN RESEARCH

A tripeptide (Gly-His-Lys) forming a stable complex with copper ions. Detected in human plasma at nanomolar concentrations; levels rise sharply at wound sites — a key endogenous signal for tissue remodelling.

— AN HONEST READING OF THE DATA

Cosmetics buried the bigger story.

Most in vivo evidence is preclinical; human skin trials exist but are small and often industry-funded.

TIER 01 / PRECLINICAL
Robust Preclinical Data
  • Collagen I & III upregulated
  • Wound closure in rodents
  • Hair follicle growth ex vivo
  • IL-6 and TNF-α reduced
  • SOD1 activation via Cu
TIER 02 / HUMAN TRIALS
Promising Skin Evidence
  • Skin elasticity improved
  • Fine lines reduced (small n)
  • Used in wound dressings
  • Hair density gains (pilot)
TIER 03 / SPECULATIVE
Emerging & Unverified
  • Neuroprotective gene effects
  • Anti-cancer gene expression
  • Systemic anti-aging claims
  • Organ protection (limited)
— GHK-CU MECHANISMS & RESEARCH DOSING READY

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— REGULATORY LANDSCAPE

GHK-Cu's Unusual Legal Position

In the UAE, research-grade peptides occupy a defined regulatory category distinct from licensed medicines. Compounds sold under this classification — including those offered by Dubai Peptides — are intended exclusively for qualified research applications, not for human administration.

GHK-Cu occupies an unusual regulatory split. Topically, it is a recognised cosmetic active — freely sold in serums and creams globally, no prescription required. That cosmetic status does not extend to injectable use. All injectable GHK-Cu on this platform is supplied as a research-grade chemical — a different product in a different regulatory category, regardless of what the topical serums on a pharmacy shelf may suggest.

1973 / DISCOVERY

Pickart identifies GHK in human plasma; patents the first copper peptide wound-healing compound.

1990s–2000s / COSMETIC ERA

GHK-Cu enters prestige skincare; ProCyte Corp licenses the compound for cosmetic wound and skin products.

2010s–PRESENT / UAE MARKET

An injectable compounding market for GHK-Cu exists in the UAE, separate from its MOHAP-listed cosmetic classification described above.